Publications

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  • 93. Application of Fragment-Based De Novo Design to the Discovery of Selective Picomolar Inhibitors of Glycogen Synthase Kinase-3 beta

    Park, S.; Shin, Y.; Kim, J.; Hong, S. 

    J. Med. Chem. 2016, 59, 9018.

  • 92. Pd(II)-Catalyzed Tandem Synthesis of Acenes Using Carboxylic Acids as Traceless Directing Groups 

    Kim, K.; Vasu, D.; Im. H.; Hong, S. 

    Angew. Chem. Int. Ed. 2016, 55, 8652. 

  • 91. Identification of Lead Small Molecule Inhibitors of Glycogen Synthase Kinase-3 beta Using a Fragment-Linking Strategy 

    Kim, J.; Moon, Y.; Hong, S.

    Bioorg. Med. Chem. Lett. 201626, 5669. 

  • 90. HS-173, a Novel PI3K Inhibitor Suppresses EMT and Metastasis in Pancreatic Cancer

    Rumman, M.; Jung, K. H.; Fang, Z.; Yan, H. H.; Son, M. K.; Kim, S. J.,; Kim, J.; Park, J. H.; Hong, S.; Hong, S.-S.

    ONCOTARGET 2016, 47, 78029. 

  • 89. Discovery of Dual Inhibitors for Wild Type and D816V Mutant of c-KIT Kinase through Virtual and Biochemical Screening of Natural Products

    Park, H.; Lee, S.; Hong, S. 

    J. Nat. Prod., 2016, 79, 293.

  • 88. Optimization and Biological Evaluation of Aminopyrimidine-based IkB Kinase b Inhibitors with Potent Anti-inflammatory Effects  

    Shin, Y.; Lim, S. M.; Yan, H. H.; Jung, S.; Fang, Z.; Jung, K. H.; Hong, S.-S.; Hong, S.

    Eur. J. Med. Chem. 2016123, 544. 

  • 87. Strategies to Overcome Acquired Resistances Conferred by Mutations in the Kinase Domain of EGFR

    Lim, S. M.; Jeong, Y.; Hong, S. 

    Future Med. Chem. 20168, 853. 

  • 86. Discovery of Low Micromolar Dual Inhibitors for Wild Type and L1196M Mutant of Anaplastic Lymphoma Kinase through the Structure-Based Virtual Screening 

    Shin, S.; Mah, S.; Hong, S.*; Park, H.* 

    J. Chem. Inf. Model. 2016, 56, 802.

  • 85. Unraveling Innate Substrate Control in Site-Selective Palladium-Catalyzed C−H Heterocycle Functionalization 

    Choi, H.; Min, M; Peng, Q.; Kang, D.; Paton, R. S.Hong, S.

    Chem. Sci. 2016, 7, 3900.  

  • 84. Rhodium-Catalyzed Direct C−H Phosphorylation of (Hetero)arenes Suitable for Late-Stage Functionalization

    Min, M.; Kang, D.; Jung, S.; Hong, S. 

    Adv. Synth. Catal., 2016, 358, 1296. (Selected as a VIP Paper by the Editorial Office.)